发明公开
EP0080695A1 Physiologically active substance FA-5859, its derivative; their production and antidiabetic agents containing said compounds
失效
生理活性化合物FA-5898，其衍生物，以及含有这些化合物的抗糖尿病剂的制备。
- 专利标题： Physiologically active substance FA-5859, its derivative; their production and antidiabetic agents containing said compounds
- 专利标题（中）： 生理活性化合物FA-5898，其衍生物，以及含有这些化合物的抗糖尿病剂的制备。
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申请号： EP82110866.9申请日： 1982-11-24
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公开(公告)号： EP0080695A1公开(公告)日： 1983-06-08
- 发明人: Kanamaru, Tsuneo , Shinagawa, Susumu , Asai, Mitsuko
- 申请人： Takeda Chemical Industries, Ltd.
- 申请人地址： 1-1, Doshomachi 4-chome Chuo-ku, Osaka JP
- 专利权人： Takeda Chemical Industries, Ltd.
- 当前专利权人： Takeda Chemical Industries, Ltd.
- 当前专利权人地址： 1-1, Doshomachi 4-chome Chuo-ku, Osaka JP
- 代理机构： von Kreisler, Alek, Dipl.-Chem.
- 优先权： PCT/JP81/00355 19811126; PCT/JP82/00291 19820728; PCT/JP82/00409 19821015
- 主分类号： C07C101/24
- IPC分类号： C07C101/24 ; C07C103/54 ; C12P13/04 ; A61K31/205
摘要：
Physiologically active substance FA-5859 and its deacetyl compound represented by the formula:
wherein R, is a hydrogen atom or an acetyl group, are produced by a cultivation of a microorganism of the genus Emericelle or Aspergillus (compound wherein R, is an acetyl group) or by a method of chemical synthesis (compound wherein R, is a hydrogen atom or an acetyl group).
Said compounds or a salt thereof have excellent fatty acid degradation inhibiting activity and is useful as an antidiabetic agent in mammalian animals or as a biochemical reagent for studies on fatty acid metabolism.
wherein R, is a hydrogen atom or an acetyl group, are produced by a cultivation of a microorganism of the genus Emericelle or Aspergillus (compound wherein R, is an acetyl group) or by a method of chemical synthesis (compound wherein R, is a hydrogen atom or an acetyl group).
Said compounds or a salt thereof have excellent fatty acid degradation inhibiting activity and is useful as an antidiabetic agent in mammalian animals or as a biochemical reagent for studies on fatty acid metabolism.
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