发明授权
- 专利标题： NOR-CHOLANIC ACID DERIVATIVES, A PROCESS FOR THEIR PREPARATION, THEIR USE AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM
- 专利标题（中）： 异丙醇酸衍生物，其制备方法，其使用和含有它们的药物组合物
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申请号： EP87900806.8申请日： 1987-01-07
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公开(公告)号： EP0253859B1公开(公告)日： 1989-05-24
- 发明人: CHIODINI, Laura , GOBBINI, Mauro , MANTEGANI, Sergio , RUGGIERI, Daniela , TEMPERILLI, Aldemio , TRAQUANDI, Gabriella , FERRARI, Patrizia
- 申请人： FARMITALIA CARLO ERBA S.r.l.
- 申请人地址： Via Carlo Imbonati 24 I-20159 Milano IT
- 专利权人： FARMITALIA CARLO ERBA S.r.l.
- 当前专利权人： FARMITALIA CARLO ERBA S.r.l.
- 当前专利权人地址： Via Carlo Imbonati 24 I-20159 Milano IT
- 代理机构： Hoffmann, Klaus, Dr. rer. nat.
- 优先权： GB8600491 19860109
- 国际公布： WO8704166 19870716
- 主分类号： C07J41/00
- IPC分类号： C07J41/00 ; A61K31/705
摘要：
Compounds (I) (either R1 = OH, C1-C4 alkoxy and R2 = H, C1-C4 alkyl, or R1 + R2 = a chemical bond; R3 = an aminodeoxy or aminodideoxy or aminotrideoxy sugar residue of the D and L series, the glycosidic linkage being alpha or beta: and either R4 = OH and R5 = H or R4 + R5 = a chemical bond) and their pharmaceutically acceptable salts are useful as antihypertensive agents. Their preparation and use as well as pharmaceutical compositions containing them are also described.
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