发明公开
EP0341462A1 Diastereoselective process for the preparation of intermediates useful for the synthesis of peptide derivatives
失效
非精神分裂症药物Verfahren zur Herstellung von Zwischenprodukten verwendbar zur Peptidderivatensynthese。
- 专利标题： Diastereoselective process for the preparation of intermediates useful for the synthesis of peptide derivatives
- 专利标题（中）： 非精神分裂症药物Verfahren zur Herstellung von Zwischenprodukten verwendbar zur Peptidderivatensynthese。
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申请号： EP89107141.7申请日： 1989-04-20
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公开(公告)号： EP0341462A1公开(公告)日： 1989-11-15
- 发明人: Pellacini, Franco , Chiarino, Dario , Carenzi, Angelo
- 申请人： ZAMBON GROUP S.p.A.
- 申请人地址： Via della Chimica, 9 I-36100 Vicenza IT
- 专利权人： ZAMBON GROUP S.p.A.
- 当前专利权人： ZAMBON GROUP S.p.A.
- 当前专利权人地址： Via della Chimica, 9 I-36100 Vicenza IT
- 优先权： IT2054288 19880511
- 主分类号： C07C227/00
- IPC分类号： C07C227/00 ; C07B53/00 ; C07C255/30
摘要：
A diastereoselective process for the preparation of compounds of formula
(wherein R and R₁ have the meanings reported in the specification and the asterisks show the asymmetric carbon atoms) starting from the corresponding N-protected 2-amino-3-aryl-propan-1-ol is described.
The compounds of formula I are intermediates useful for the synthesis of pharmacologically active peptides.
(wherein R and R₁ have the meanings reported in the specification and the asterisks show the asymmetric carbon atoms) starting from the corresponding N-protected 2-amino-3-aryl-propan-1-ol is described.
The compounds of formula I are intermediates useful for the synthesis of pharmacologically active peptides.
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