发明公开
EP1414806A1 NOVEL VINYL N-(2-BENZOYLPHENYL)-L-TYROSINE DERIVATIVES AND THEIR USE AS ANTIDIABETICS ETC
审中-公开
NEW VINYL-N-（2-苯甲酰基苯基）-L-酪氨酸衍生物及其作为抗糖尿病ETC.
- 专利标题： NOVEL VINYL N-(2-BENZOYLPHENYL)-L-TYROSINE DERIVATIVES AND THEIR USE AS ANTIDIABETICS ETC
- 专利标题（中）： NEW VINYL-N-（2-苯甲酰基苯基）-L-酪氨酸衍生物及其作为抗糖尿病ETC.
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申请号： EP02745184.8申请日： 2002-07-05
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公开(公告)号： EP1414806A1公开(公告)日： 2004-05-06
- 发明人: JEPPESEN, Lone , BURY, Paul, Stanley , MOGENSEN, John, Patrick , PETTERSSON, Ingrid , SAUERBERG, Per
- 申请人： NOVO NORDISK A/S
- 申请人地址： Novo Allé 2880 Bagsvaerd DK
- 专利权人： NOVO NORDISK A/S
- 当前专利权人： NOVO NORDISK A/S
- 当前专利权人地址： Novo Allé 2880 Bagsvaerd DK
- 代理机构： Madsen, Inger Margrethe Schelde
- 优先权： DK200101156 20010730
- 国际公布： WO2003011834 20030213
- 主分类号： C07D235/16
- IPC分类号： C07D235/16 ; C07D279/22 ; C07D471/04 ; C07D209/86 ; C07D223/22 ; A61K31/538 ; A61K31/5415 ; A61K31/403 ; A61K31/55 ; A61P1/18 ; A61P3/06 ; A61P3/10
摘要：
Novel compounds of the general formula (I), the use of these compounds as medicaments, pharmaceutical compositions comprising the compounds and methods of treatment employing these compounds and compositions. The present compounds may be useful in the treatment and/or prevention of conditions mediated by nuclear receptors, in particular the Peroxisome Proliferator-Activated Receptors (PPAR). The compounds exert their effects by modulating the PPARη response in a partial agonist manner.
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