发明公开
- 专利标题： NEW METHIONINE AMINOPEPTIDASE INHIBITOR
- 专利标题（中）： 中性甲硫氨酸氨基转移酶抑制剂
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申请号： EP03711802.3申请日： 2003-03-25
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公开(公告)号： EP1500655A1公开(公告)日： 2005-01-26
- 发明人: NAN, Fajun, The National Center For Drug Screening , YE, Qizhuang, The National Center For Drug Screen. , LI, Jingya, The National Center For Drug Screening , LIU, Zhiying, The National Center For Drug Screen. , LUO, Qunli, The National Center For Drug Screening , CUI, Yongmei, The National Center For Drug Screen.
- 申请人： Shanghai Institute of Materia Medica, Chinese Academy of Sciences
- 申请人地址： 555 Zu Chong Zhi Road Pudong New, Shanghai 201203 CN
- 专利权人： Shanghai Institute of Materia Medica, Chinese Academy of Sciences
- 当前专利权人： Shanghai Institute of Materia Medica, Chinese Academy of Sciences
- 当前专利权人地址： 555 Zu Chong Zhi Road Pudong New, Shanghai 201203 CN
- 代理机构： Epping Hermann & Fischer
- 优先权： CN02111230 20020402
- 国际公布： WO2003082838 20031009
- 主分类号： C07D277/22
- IPC分类号： C07D277/22 ; C07D277/38 ; C07D263/30 ; C07D263/48 ; C07D207/30 ; C07D207/34 ; C07D401/12 ; C07D403/12 ; C07D405/12 ; C07D407/12 ; C07D417/12 ; A61K31/40 ; A61K31/41
摘要：
The invention provides a new methionine aminopeptidase inhibitors with the following formula (I), wherein R 1 , R 2 , R 3 , R 4 , R 5 , R 6 and X have the meanings given in the description. Pharmacological experiment shows that they display good inhibition activity for methionine aminopeptidase.
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