发明公开
- 专利标题： CYCLOPROPYL BETA-AMINO ACID DERIVATIVES
- 专利标题（中）： 环丙基BETA-AMINOSÄUREDERIVATE
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申请号： EP04701059.0申请日： 2004-01-09
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公开(公告)号： EP1592661A2公开(公告)日： 2005-11-09
- 发明人: SCHWARZ, Jacob Bradley,Pfizer Global Res. & Dev. , WUSTROW, David Juergen,Pfizer Global Res. & Dev.
- 申请人： Warner-Lambert Company LLC
- 申请人地址： 201 Tabor Road Morris Plains,New Jersey 07950 US
- 专利权人： Warner-Lambert Company LLC
- 当前专利权人： Warner-Lambert Company LLC
- 当前专利权人地址： 201 Tabor Road Morris Plains,New Jersey 07950 US
- 代理机构： Cosway, Sarah Michelle
- 优先权： US441825P 20030122
- 国际公布： WO2004065361 20040805
- 主分类号： C07D201/00
- IPC分类号： C07D201/00
摘要：
This invention relates to novel cyclopropyl β-amino acids derivatives of the formula (I) wherein R1 through R4 are defined as in the specification, pharmaceutical compositions containing them and their use for the treatment of various central nervous system and other disorders. The cyclopropyl β-amino acids derivatives of this invention exhibit activity as alpha2delta ligands (α2δ ligands). Such compounds have affinity for the α2δ subunit of a calcium channel.
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