发明公开
EP1717233A1 Histamine H3-receptor ligands and their therapeutic application
审中-公开
Ligandenfürden Histamin H3-Rezeptor und ihre therapeutische Anwendung
- 专利标题： Histamine H3-receptor ligands and their therapeutic application
- 专利标题（中）： Ligandenfürden Histamin H3-Rezeptor und ihre therapeutische Anwendung
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申请号： EP05290948.8申请日： 2005-04-29
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公开(公告)号： EP1717233A1公开(公告)日： 2006-11-02
- 发明人: Bertrand, Isabelle , Capet, Marc , Lecomte, Jeanne-Marie , Levoin, Nicolas , Ligneau,Xavier , Poupardin-Olivier, Olivia , Robert, Philippe , Schwartz, Jean-Charles
- 申请人： BIOPROJET
- 申请人地址： 30, rue des Francs-Bourgeois 75003 Paris FR
- 专利权人： BIOPROJET
- 当前专利权人： BIOPROJET
- 当前专利权人地址： 30, rue des Francs-Bourgeois 75003 Paris FR
- 代理机构： Colombet, Alain André
- 主分类号： C07D295/088
- IPC分类号： C07D295/088 ; C07D307/79 ; C07D317/54 ; C07D319/18 ; A61K31/40 ; A61K31/445 ; A61P25/00
摘要：
The present patent application concerns new compounds of formula (I)
with R 1 and R 2 taken together with the nitrogen atom to which they are attached, form a saturated nitrogen-containing ring, A is a saturated C1-4 alkylene and B a C3-4 alkylene or alkenylene chain; their preparation and their use as a H3 receptor ligand for treating e.g. CNS disorders like Alzheimer's disease.
with R 1 and R 2 taken together with the nitrogen atom to which they are attached, form a saturated nitrogen-containing ring, A is a saturated C1-4 alkylene and B a C3-4 alkylene or alkenylene chain; their preparation and their use as a H3 receptor ligand for treating e.g. CNS disorders like Alzheimer's disease.
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