发明公开
- 专利标题： AMINOPHENYLSULFONAMIDE DERIVATIVES AS HIV PROTEASE INHIBITOR
- 专利标题（中）： 作为HIV蛋白酶抑制剂的氨基苯磺酰胺衍生物
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申请号： EP06819805.0申请日： 2006-11-28
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公开(公告)号： EP1960381A1公开(公告)日： 2008-08-27
- 发明人: DE KOCK, Herman Augustinus , JONCKERS, Tim Hugo Maria , LAST, Stefaan Julien , BOONANTS, Paul Jozef Gabriel Maria , SURLERAUX, Dominique Louis Nestor Ghislain , WIGERINCK, Piet Tom Bert Paul
- 申请人： Tibotec Pharmaceuticals Ltd.
- 申请人地址： Eastgate Village Eastgate Little Island Co Cork IE
- 专利权人： Tibotec Pharmaceuticals Ltd.
- 当前专利权人： Tibotec Pharmaceuticals Ltd.
- 当前专利权人地址： Eastgate Village Eastgate Little Island Co Cork IE
- 代理机构： Daelemans, Frank F.R.
- 优先权： EP05111393 20051128
- 国际公布： WO2007060249 20070531
- 主分类号： C07D401/04
- IPC分类号： C07D401/04 ; A61K31/34 ; A61P31/18
摘要：
The present invention concerns substituted aminophenylsulfonamide compounds and derivatives, their use as protease inhibitors, in particular as broadspectrum HIV protease inhibitors, processes for their preparation as well as pharmaceutical compositions and diagnostic kits comprising them. The present invention also concerns combinations of the present substituted aminophenylsulfonamide compounds and derivatives with another anti-retroviral agent. It further relates to their use in assays as reference compounds or as reagents.
公开/授权文献
- EP1960381B1 AMINOPHENYLSULFONAMIDE DERIVATIVES AS HIV PROTEASE INHIBITOR 公开/授权日：2015-06-17
信息查询
