发明公开
EP2440533A1 GUANINE RIBOSWITCH BINDING COMPOUNDS AND THEIR USE AS ANTIBIOTICS
有权
鸟嘌呤核糖开关结合的化合物及其用途抗生素
- 专利标题： GUANINE RIBOSWITCH BINDING COMPOUNDS AND THEIR USE AS ANTIBIOTICS
- 专利标题（中）： 鸟嘌呤核糖开关结合的化合物及其用途抗生素
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申请号： EP10785625.4申请日： 2010-06-14
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公开(公告)号： EP2440533A1公开(公告)日： 2012-04-18
- 发明人: MULHBACHER, Jérôme , LAFONTAINE , Daniel , MALOUIN , François , ALLARD , Marianne , MARSAULT , Eric
- 申请人： Socpra-Sciences Et Génie S.E.C.
- 申请人地址： Suite 100, 35 rue Radisson Sherbrooke, Québec J1L 1E2 CA
- 专利权人： Socpra-Sciences Et Génie S.E.C.
- 当前专利权人： Socpra-Sciences Et Génie S.E.C.
- 当前专利权人地址： Suite 100, 35 rue Radisson Sherbrooke, Québec J1L 1E2 CA
- 代理机构： Ilgart, Jean-Christophe
- 优先权： US186669P 20090612; US307088P 20100223
- 国际公布： WO2010142027 20101216
- 主分类号： C07D239/46
- IPC分类号： C07D239/46 ; A61K31/513 ; A61K31/519 ; A61L2/16 ; A61P31/04 ; C07D239/48 ; C07D239/50 ; C07D239/56 ; C07D498/04 ; C07D513/04 ; G01N33/569
摘要：
The present invention includes novel compounds and pharmaceutically acceptable formulations of said compounds which exhibit antibiotic activity against microorganisms bearing a guanine riboswitch that controls the expression of the guaA gene, including organisms which are resistant to certain antibiotic families, and which are useful as antibacterial agents for treatment or prophylaxis of bacterial infections in animals or in humans, in particular but not limited to infections of the mammary gland, or their use as antiseptics, agents for sterilization or disinfection.
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