发明公开
EP2476683A2 NOVEL TETRA-AZA MACROCYCLIC COMPOUND, METHOD FOR PREPARING SAME, AND USE THEREOF
审中-公开
NEER MAKROZYKLISCHE TETRA-AZA-VERBINDUNG，VERFAHREN ZU IHRER HERSTELLUNG UND VERWENDUNG DAVON
- 专利标题： NOVEL TETRA-AZA MACROCYCLIC COMPOUND, METHOD FOR PREPARING SAME, AND USE THEREOF
- 专利标题（中）： NEER MAKROZYKLISCHE TETRA-AZA-VERBINDUNG，VERFAHREN ZU IHRER HERSTELLUNG UND VERWENDUNG DAVON
-
申请号： EP10815618.3申请日： 2010-09-09
-
公开(公告)号： EP2476683A2公开(公告)日： 2012-07-18
- 发明人: YOO, Jeong Soo , PANDYA, Darpan
- 申请人： Kyungpook National University Industry- Academic Cooperation Foundation
- 申请人地址： Kyungpook National University 1370 Sangyeok-dong Buk-gu Daegu 702-701 KR
- 专利权人： Kyungpook National University Industry- Academic Cooperation Foundation
- 当前专利权人： Kyungpook National University Industry- Academic Cooperation Foundation
- 当前专利权人地址： Kyungpook National University 1370 Sangyeok-dong Buk-gu Daegu 702-701 KR
- 代理机构： Ehnis, Tobias
- 优先权： KR20090084943 20090909; KR20100073954 20100730
- 国际公布： WO2011031073 20110317
- 主分类号： C07D487/04
- IPC分类号： C07D487/04 ; C07D403/12 ; C07D257/02 ; A61K49/04 ; A61P35/00 ; A61P31/00
摘要：
Provided are a cross-bridged tetraaza macrocyclic compound of a novel structure that can be used, for example, as a contrast agent for diagnostic imaging or a radiopharmaceutical and a method for preparing the same.
The disclosed tetraaza macrocyclic compound is able to form a stable metal complex at a lower temperature and allows easy conjugation with a bioactive substance or a chemically active substance, when compared to the existing cross-bridged tetraaza macrocyclic compounds.
The disclosed tetraaza macrocyclic compound is able to form a stable metal complex at a lower temperature and allows easy conjugation with a bioactive substance or a chemically active substance, when compared to the existing cross-bridged tetraaza macrocyclic compounds.
公开/授权文献
信息查询
