发明公开
EP2760871A1 OXY-CYCLOHEXYL-4H,6H-5-OXA-2,3,10B-TRIAZA-BENZO[E]AZULENES AS V1A ANTAGONISTS
有权
OXY-CYCLOHEXYL-4H，6H-5-OXA-2,3,10B-三唑 - 苯并[E]亚油酸乙酯V1A-ANTAGONISTEN
- 专利标题： OXY-CYCLOHEXYL-4H,6H-5-OXA-2,3,10B-TRIAZA-BENZO[E]AZULENES AS V1A ANTAGONISTS
- 专利标题（中）： OXY-CYCLOHEXYL-4H，6H-5-OXA-2,3,10B-三唑 - 苯并[E]亚油酸乙酯V1A-ANTAGONISTEN
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申请号： EP12761740.5申请日： 2012-09-24
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公开(公告)号： EP2760871A1公开(公告)日： 2014-08-06
- 发明人: DOLENTE, Cosimo , SCHNIDER, Patrick
- 申请人： F.Hoffmann-La Roche AG
- 申请人地址： Grenzacherstrasse 124 4070 Basel CH
- 专利权人： F.Hoffmann-La Roche AG
- 当前专利权人： F.Hoffmann-La Roche AG
- 当前专利权人地址： Grenzacherstrasse 124 4070 Basel CH
- 代理机构： Müller-Afraz, Simona
- 优先权： EP11182796 20110926
- 国际公布： WO2013045373 20130404
- 主分类号： C07D498/04
- IPC分类号： C07D498/04 ; A61K31/553 ; A61P9/12
摘要：
The present invention provides 4H,6H-5-oxa-2,3,10b-triaza-benzo[e]azulenes of the formula wherein R1 and R2 are as defined herein and which act as V1a receptor modulators, and in particular as V1a receptor antagonists, their manufacture, pharmaceutical compositions containing them and their use as medicaments.
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