发明公开
EP2834229A1 PROCESS FOR THE MANUFACTURING OF CCR3 INHIBITORS
有权
VERFAHREN ZUR HERSTELLUNG VON CCR3-INHIBITOREN
- 专利标题： PROCESS FOR THE MANUFACTURING OF CCR3 INHIBITORS
- 专利标题（中）： VERFAHREN ZUR HERSTELLUNG VON CCR3-INHIBITOREN
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申请号： EP13712567.0申请日： 2013-03-28
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公开(公告)号： EP2834229A1公开(公告)日： 2015-02-11
- 发明人: DURAN, Adil , SCHMID, Rolf
- 申请人： Boehringer Ingelheim International GmbH
- 申请人地址： Binger Strasse 173 55216 Ingelheim am Rhein DE
- 专利权人： Boehringer Ingelheim International GmbH
- 当前专利权人： Boehringer Ingelheim International GmbH
- 当前专利权人地址： Binger Strasse 173 55216 Ingelheim am Rhein DE
- 代理机构： Simon, Elke Anna Maria
- 优先权： EP12162852 20120402
- 国际公布： WO2013149926 20131010
- 主分类号： C07D401/12
- IPC分类号： C07D401/12
摘要：
The present invention relates to a process for preparing CCR3 inhibitors of formula (1), wherein R
1 is H, C
1-6 -alkyl, C
0-4 -alkyl-C
3-6 -cycloalkyl, C
1-6 -haloalkyl; R
2 is H, C
1-6 -alkyl; Xis an anion selected from the group consisting of chloride or ½ dibenzoyltartrate; j is 1 or 2.
1 is H, C
1-6 -alkyl, C
0-4 -alkyl-C
3-6 -cycloalkyl, C
1-6 -haloalkyl; R
2 is H, C
1-6 -alkyl; Xis an anion selected from the group consisting of chloride or ½ dibenzoyltartrate; j is 1 or 2.
公开/授权文献
- EP2834229B1 PROCESS FOR THE MANUFACTURING OF CCR3 INHIBITORS 公开/授权日：2017-08-09
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