发明公开
EP3109245A4 METHOD FOR PRODUCTING THIOLANE SKELETON-TYPE GLYCOCONJUGATE, AND THIOLANE SKELETON-TYPE GLYCOCONJUGATE
有权
VERFAHREN ZUR HERSTELLUNG EINES THIOLANSKELETTARTIGEN GLYCOKONJUGATS UND THIOLANSKELETTARTIGES GLYCOKONJUGAT
- 专利标题: METHOD FOR PRODUCTING THIOLANE SKELETON-TYPE GLYCOCONJUGATE, AND THIOLANE SKELETON-TYPE GLYCOCONJUGATE
- 专利标题(中): VERFAHREN ZUR HERSTELLUNG EINES THIOLANSKELETTARTIGEN GLYCOKONJUGATS UND THIOLANSKELETTARTIGES GLYCOKONJUGAT
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申请号: EP15751503申请日: 2015-02-17
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公开(公告)号: EP3109245A4公开(公告)日: 2017-03-01
- 发明人: ITO TAKAYUKI , WATANABE TORU , OKADA HIDEKI , KUNIYOSHI HIDENOBU
- 申请人: FUJIFILM CORP
- 专利权人: FUJIFILM CORP
- 当前专利权人: FUJIFILM CORP
- 优先权: JP2014029020 2014-02-18; JP2014220368 2014-10-29
- 主分类号: C07H1/00
- IPC分类号: C07H1/00 ; C07D333/32 ; C07H13/08 ; C07H15/04 ; C07H15/18
摘要:
There is provided a production method of a compound represented by the following formula (II) through a step of reacting a compound represented by the following General Formula (I) with a sulfur compound. In General Formulas (I) and (II), R 1 represents a hydrogen atom or an acyl group, R 2 represents a hydrogen atom, a fluorine atom, an acyloxy group, an arylmethyloxy group, an allyloxy group, an arylmethyloxycarbonyloxy group, or an allyloxycarbonyloxy group, R 3 represents a hydrogen atom or an acyloxy group, R 5 represents an alkyl group or an aryl group, and X represents a leaving group. Here, in a case where R 2 is a fluorine atom, an acyloxy group, an arylmethyloxy group, an allyloxy group, an arylmethyloxycarbonyloxy group, or an allyloxycarbonyloxy group, R 3 is an acyloxy group.
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