发明公开
- 专利标题： PYRIDYL OR PYRAZINYL COMPOUNDS CARRYING A METHYL-BOUND ALPHA-AMINO ACID AMIDE GROUP
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申请号： EP16770000.4申请日： 2016-09-21
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公开(公告)号： EP3353155A1公开(公告)日： 2018-08-01
- 发明人: BACKFISCH, Gisela , BAKKER, Margaretha , BLAICH, Günter , BRAJE, Wilfried , DRESCHER, Karla , ERHARD, Thomas , HAUPT, Andreas , HOFT, Carolin , KLING, Andreas , LAKICS, Viktor , MACK, Helmut , OELLIEN, Frank , PETER, Raimund , POHLKI, Frauke , RELO, Ana Lucia
- 申请人： AbbVie Deutschland GmbH & Co. KG
- 申请人地址： Mainzer Strasse 81 65189 Wiesbaden DE
- 专利权人： AbbVie Deutschland GmbH & Co. KG
- 当前专利权人： AbbVie Deutschland GmbH & Co. KG
- 当前专利权人地址： Mainzer Strasse 81 65189 Wiesbaden DE
- 代理机构： Reitstötter Kinzebach
- 优先权： US201562221350P 20150921
- 国际公布： WO2017050807 20170330
- 主分类号： C07D241/20
- IPC分类号： C07D241/20 ; C07D213/56 ; A61K31/4439 ; A61K31/497 ; A61P25/00
摘要：
The present invention relates to pyridyl or pyrazinyl compounds carrying a methyl- bound N-amide moiety derived from an α-amino acid of formula I where the variables are as defined in the claims and the description. The invention further relates to a pharmaceutical composition containing such compounds, to their use as modulators, especially agonists or partial agonists, of the 5-HT2C receptor, and to their use for preparing a medicament for the prevention or treatment of conditions and disorders which respond to the modulation of the 5-HT2C receptor.
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