- 专利标题: METHOD FOR THE SYNTHESIS OF CYCLIC DEPSIPEPTIDES
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申请号: EP17200415.2申请日: 2017-11-07
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公开(公告)号: EP3480195A1公开(公告)日: 2019-05-08
- 发明人: The designation of the inventor has not yet been filed
- 申请人: Bayer Animal Health GmbH , The Kitasato Institute
- 申请人地址: Kaiser-Wilhelm-Allee 10 51373 Leverkusen DE
- 专利权人: Bayer Animal Health GmbH,The Kitasato Institute
- 当前专利权人: Bayer Animal Health GmbH,The Kitasato Institute
- 当前专利权人地址: Kaiser-Wilhelm-Allee 10 51373 Leverkusen DE
- 代理机构: BIP Patents
- 主分类号: C07D413/14
- IPC分类号: C07D413/14 ; A01N43/72 ; A61K38/15 ; A61K45/06 ; C07C269/06 ; C07C271/22 ; C07B51/00 ; C07C231/12 ; C07D273/00 ; C07D273/08 ; C07K11/02
摘要:
The present invention relates to a method for the synthesis of cyclic depsipeptides, in particular emodepside, involving specific carboxylic acid group protecting tags:
TAG is preferably:
wherein m is ≥ 15 to ≤ 25, p is ≥ 8 to ≤ 18 and q is ≥ 15 to ≤ 25.
TAG is preferably:
wherein m is ≥ 15 to ≤ 25, p is ≥ 8 to ≤ 18 and q is ≥ 15 to ≤ 25.
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