Invention Grant
- Patent Title: 5-substituted-5-hydroxy-5-aryl-3-oxo-pentanoate derivatives and their enantiopure forms
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Application No.: US15560868Application Date: 2016-02-01
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Publication No.: US10125074B2Publication Date: 2018-11-13
- Inventor: Fujie Tanaka , Dongxin Zhang
- Applicant: OKINAWA INSTITUTE OF SCIENCE AND TECHNOLOGY SCHOOL CORPORATION
- Applicant Address: JP Okinawa
- Assignee: OKINAWA INSTITUTE OF SCIENCE AND TECHNOLOGY SCHOOL CORPORATION
- Current Assignee: OKINAWA INSTITUTE OF SCIENCE AND TECHNOLOGY SCHOOL CORPORATION
- Current Assignee Address: JP Okinawa
- Agency: Wenderoth, Lind & Ponack, L.L.P.
- Priority: JP2015-152438 20150731
- International Application: PCT/JP2016/000507 WO 20160201
- International Announcement: WO2016/151990 WO 20160929
- Main IPC: C07C49/00
- IPC: C07C49/00 ; C07C69/00 ; C07C227/30 ; C07C49/753 ; C07C69/738 ; C07D333/22 ; C07D333/24 ; C07C227/10 ; C07C229/34 ; C07C49/255 ; C07C49/747 ; C07C227/34 ; C07C227/42 ; A61K31/02 ; A61K31/045
Abstract:
The present invention relates to novel tertiary alcohol derivatives substituted with aryl and trifluoromethyl, and optical isomers thereof. In addition, the present invention also relates to methods for the preparation and use as enantiomer recognition agent thereof. The present invention provides pharmaceutical composition and use as therapeutically active substance thereof.
Public/Granted literature
- US20180118648A1 5-SUBSTITUTED-5-HYDROXY-5-ARYL-3-OXO-PENTANOATE DERIVATIVES AND THEIR ENANTIOPURE FORMS Public/Granted day:2018-05-03
Information query
