- 专利标题: Tricyclic benzoxaborole compounds and uses thereof
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申请号: US15792251申请日: 2017-10-24
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公开(公告)号: US10308668B2公开(公告)日: 2019-06-04
- 发明人: Michael Richard Kevin Alley , Vincent Hernandez , Jacob J. Plattner , Xianfeng Li , David Barros-Aguirre , Ilaria Giordano
- 申请人: GLAXOSMITHKLINE INTELLECTUAL PROPERTY (NO.2) LIMITED , ANACOR PHARMACEUTICALS INC.
- 申请人地址: GB Brentford, Middlesex CA Palo Alto
- 专利权人: GlaxoSmithKline Intellectual Property (No. 2) Limited,Anacor Pharmaceuticals, Inc.
- 当前专利权人: GlaxoSmithKline Intellectual Property (No. 2) Limited,Anacor Pharmaceuticals, Inc.
- 当前专利权人地址: GB Brentford, Middlesex CA Palo Alto
- 代理机构: Dority & Manning, P.A.
- 主分类号: C07F5/02
- IPC分类号: C07F5/02 ; A61K31/69 ; C07F5/04 ; A61K45/06
摘要:
Compounds of Formula II, wherein X is selected from chloro, fluoro, bromo and iodo, R1 and R2 are each independently selected from H, —CH3, —CH2CH3, —CH2CH2CH3, or —CH(CH3)2; compositions containing them, their use in therapy, including their use as anti-mycobacterial agents, for example in the treatment of a mycobacterial infection in a mammal, and methods for the preparation of such compounds, are provided.
公开/授权文献
- US20180044355A1 TRICYCLIC BENZOXABOROLE COMPOUNDS AND USES THEREOF 公开/授权日:2018-02-15