- 专利标题： Pyridinone dicarboxamide for use as bromodomain inhibitors
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申请号： US15762229申请日： 2016-09-20
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公开(公告)号： US10370356B2公开(公告)日： 2019-08-06
- 发明人: Stephen John Atkinson , Emmanuel Hubert Demont , Lee Andrew Harrison , Thomas George Christopher Hayhow , David House , Matthew J. Lindon , Alexander G. Preston , Jonathan Thomas Seal , Ian David Wall , Robert J. Watson , James Michael Woolven
- 申请人： GlaxoSmithKline Intellectual Property (No. 2) Limited
- 申请人地址： GB Brentford, Middlesex
- 专利权人： GlaxoSmithKline Intellectual Property (No. 2) Limited
- 当前专利权人： GlaxoSmithKline Intellectual Property (No. 2) Limited
- 当前专利权人地址： GB Brentford, Middlesex
- 代理商 Jane F. Djung; Duke M. Fitch; Edward R. Gimmi
- 国际申请： PCT/EP2016/072216 WO 20160920
- 国际公布： WO2017/050714 WO 20170330
- 主分类号： C07D401/12
- IPC分类号： C07D401/12 ; C07D401/14 ; C07D405/12 ; C07D409/12 ; A61K31/4427 ; A61K31/443 ; A61K31/4433 ; A61K31/4436 ; A61K31/4545 ; A61K31/496 ; A61K31/5377 ; A61K31/541
摘要：
The present invention relates to compounds of formula (I) and salts thereof, pharmaceutical compositions containing such compounds and to their use in therapy