Invention Grant
- Patent Title: Methyl 2-methyl-5-oxo-1,4,5,7-tetradhydrofuro[3,4-b]pyridine-3-carboxylate compounds as Cav1.2 activators
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Application No.: US17345902Application Date: 2021-06-11
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Publication No.: US11453679B2Publication Date: 2022-09-27
- Inventor: Thomas Charles Caya , James Neef , Tejaskumar Pankajbhai Pathak , Amir Masoud Sadaghiani , Xilin Zhou
- Applicant: Novartis AG
- Applicant Address: CH Basel
- Assignee: Novartis AG
- Current Assignee: Novartis AG
- Current Assignee Address: CH Basel
- Agency: Finnegan, Henderson, Farabow, Garrett & Dunner, LLP
- Main IPC: C07D491/048
- IPC: C07D491/048
![Methyl 2-methyl-5-oxo-1,4,5,7-tetradhydrofuro[3,4-b]pyridine-3-carboxylate compounds as Cav1.2 activators](/abs-image/US/2022/09/27/US11453679B2/abs.jpg.150x150.jpg)
Abstract:
The present disclosure provides for a compound according to formula (I) or a pharmaceutically acceptable salt thereof as Cav1.2 activators for the treatment of schizophrenia, bipolar disorder, major depressive disorder, substance use disorder, ADHD, Phelan-McDermid Syndrome, autism spectrum disorder, multiple sclerosis, frontotemporal dementia, Alzheimer's disease, Brugada Syndrome, Short QT syndrome, and early repolarization syndrome.
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