发明申请
US20050065146A1 Novel benzothiazine and benzothiadiazine derivatives, method for preparing same and pharmaceutical compositions containing same
失效
新的苯并噻嗪和苯并噻二嗪衍生物，其制备方法和含有它们的药物组合物
- 专利标题： Novel benzothiazine and benzothiadiazine derivatives, method for preparing same and pharmaceutical compositions containing same
- 专利标题（中）： 新的苯并噻嗪和苯并噻二嗪衍生物，其制备方法和含有它们的药物组合物
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申请号： US10499164申请日： 2002-12-20
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公开(公告)号： US20050065146A1公开(公告)日： 2005-03-24
- 发明人: Alex Cordi , Patrice Desos , Pierre Lestage
- 申请人： Alex Cordi , Patrice Desos , Pierre Lestage
- 优先权： FR01/16620 20011221
- 国际申请： PCT/FR02/04483 WO 20021220
- 主分类号： C07D285/24
- IPC分类号： C07D285/24 ; A61K31/549 ; A61P25/00 ; A61P25/08 ; A61P25/14 ; A61P25/18 ; A61P25/22 ; A61P25/24 ; A61P25/28 ; C07D279/02 ; C07D513/04 ; C07D498/04
摘要：
Compounds of formula (I): wherein: R1 represents aryl or heteroaryl, R2 represents hydrogen, halogen or hydroxy, X represents oxygen or sulphur, Y represents oxygen, sulphur or NR wherein R represents hydrogen or alkyl, A represents CR4R5 or NR4, R3 represents hydrogen, alkyl or cycloalkyl, R4 represents hydrogen or alkyl, or A represents nitrogen and, together with adjacent —CHR3—, forms the ring wherein m represents 1, 2 or 3, R5 represents hydrogen or halogen, their isomers and also their addition salts Medicaments.