发明申请
US20050113309A1 Crystalline forms(2s)-n-5[amino(imino)methyl]-2-thienylmethyl-1-(2r)-2[(carboxymethyl) amino]-3,3-diphenylpropanoyl-2-pyrrolidinecarboxamide nh2o
审中-公开
结晶形式(2s)-n-5 [氨基(亚氨基)甲基] -2-噻吩甲基-1-(2r)-2 [(羧甲基)氨基] -3,3-二苯基丙酰基-2-吡咯烷甲酰胺nh2o
- 专利标题: Crystalline forms(2s)-n-5[amino(imino)methyl]-2-thienylmethyl-1-(2r)-2[(carboxymethyl) amino]-3,3-diphenylpropanoyl-2-pyrrolidinecarboxamide nh2o
- 专利标题(中): 结晶形式(2s)-n-5 [氨基(亚氨基)甲基] -2-噻吩甲基-1-(2r)-2 [(羧甲基)氨基] -3,3-二苯基丙酰基-2-吡咯烷甲酰胺nh2o
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申请号: US10508524申请日: 2003-03-21
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公开(公告)号: US20050113309A1公开(公告)日: 2005-05-26
- 发明人: Aeri Kim , Jae-Hyeon Park , Suk-Kyoon Yoon , Bong-Chan Kim , Sung-Ji Kim , Kwan-Hyung Cho
- 申请人: Aeri Kim , Jae-Hyeon Park , Suk-Kyoon Yoon , Bong-Chan Kim , Sung-Ji Kim , Kwan-Hyung Cho
- 优先权: KR10-2002-0015627 20020322
- 国际申请: PCT/KR03/00558 WO 20030321
- 主分类号: A61K38/00
- IPC分类号: A61K38/00 ; A61P7/02 ; C07D409/12 ; C07K5/06 ; C07K5/065 ; A61K38/04 ; A61K31/4025 ; C07D49/02
摘要:
The present invention relates to crystalline forms of (2S)-N-5-[amino(imino)methyl]-2-thienyl-methyl-1-(2R)-2-[(carboxymethyl)amino]-3,3-diphenylpropanoyl-2-pyrrolidinecarboxamide nH2O.