发明申请
US20050124606A1 Novel benzothiazine and benzothiadiazine derivatives method for preparing same and pharmaceutical compositions containing same
失效
新颖的苯并噻嗪和苯并噻二嗪衍生物的制备方法和含有它们的药物组合物
- 专利标题: Novel benzothiazine and benzothiadiazine derivatives method for preparing same and pharmaceutical compositions containing same
- 专利标题(中): 新颖的苯并噻嗪和苯并噻二嗪衍生物的制备方法和含有它们的药物组合物
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申请号: US10498948申请日: 2002-12-20
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公开(公告)号: US20050124606A1公开(公告)日: 2005-06-09
- 发明人: Alex Cordi , Patrice Desos , Pierre Lestage
- 申请人: Alex Cordi , Patrice Desos , Pierre Lestage
- 优先权: FR01/16621 20011221
- 国际申请: PCT/FR02/04485 WO 20021220
- 主分类号: C07D285/24
- IPC分类号: C07D285/24 ; A61K31/549 ; A61K31/662 ; A61P9/10 ; A61P25/00 ; A61P25/08 ; A61P25/14 ; A61P25/18 ; A61P25/22 ; A61P25/24 ; A61P25/28 ; A61P43/00 ; C07D279/02 ; C07D417/12 ; C07D513/04 ; C07D498/14
摘要:
Compounds of formula (I): wherein: R1 represents aryl or heteroaryl, R2 represents hydrogen, halogen or hydroxy, A represents CR4R5 or NR4, R3 represents hydrogen, alkyl or cycloalkyl, R4 represents hydrogen or alkyl, or A represents nitrogen and, together with adjacent —CHR3—, forms the ring wherein m represents 1, 2 or 3, R5 represents hydrogen or halogen, their isomers and also their addition salts. Medicaments.
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