发明申请
US20050245553A1 Methods of treating medical conditions using sulfonate-substituted pyrazolopyridine derivatives
失效
使用磺酸酯取代的吡唑并吡啶衍生物治疗医学病症的方法
- 专利标题： Methods of treating medical conditions using sulfonate-substituted pyrazolopyridine derivatives
- 专利标题（中）： 使用磺酸酯取代的吡唑并吡啶衍生物治疗医学病症的方法
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申请号： US11175740申请日： 2005-07-05
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公开(公告)号： US20050245553A1公开(公告)日： 2005-11-03
- 发明人: Johannes-Peter Stasch , Achim Feurer , Stefan Weigand , Elke Stahl , Dietmar Flubacher , Cristina Alonso-Alija , Frank Wunder , Dieter Lang , Klaus Dembowsky , Alexander Straub , Elisabeth Perzborn
- 申请人： Johannes-Peter Stasch , Achim Feurer , Stefan Weigand , Elke Stahl , Dietmar Flubacher , Cristina Alonso-Alija , Frank Wunder , Dieter Lang , Klaus Dembowsky , Alexander Straub , Elisabeth Perzborn
- 申请人地址： DE Leverkusen
- 专利权人： Bayer Aktiengesellschaft
- 当前专利权人： Bayer Aktiengesellschaft
- 当前专利权人地址： DE Leverkusen
- 优先权： DE10122894.5 20010511
- 主分类号： A61K31/506
- IPC分类号： A61K31/506 ; A61K45/00 ; A61P9/00 ; A61P9/10 ; A61P9/12 ; A61P15/10 ; A61P25/00 ; A61P29/00 ; C07D471/04 ; A61K31/513 ; C07D471/02
摘要：
This invention relates to methods of treatment of cardiovascular disorders, thromboembolic disorders, inflammation, and disorders of the central nervous system using pyrazol pyridine derivatives of formula (I) wherein R1 is a radical of the formula —O—SO2-R3 in which R3 is optionally substituted C1-6-alkyl, optionally substituted C3-8-cycloalkyl, or optionally substituted phenyl; R2 is H, optionally substituted C1-6-alkyl-CO— or optionally substituted C1-6-alkyl-SO2—; as well as salts, stereoisomers, tautomers, and hydrates thereof.