发明申请
US20050272749A1 5-Alkyl-7-aminotriazolopyrimidines, methods and intermediary product necessary for the production thereof, agents containing said compounds and the use thereof for fighting against harmful mushrooms
失效
5-烷基-7-氨基三唑并嘧啶，其生产所需的方法和中间产物，含有所述化合物的试剂及其用于防治有害蘑菇的用途
- 专利标题： 5-Alkyl-7-aminotriazolopyrimidines, methods and intermediary product necessary for the production thereof, agents containing said compounds and the use thereof for fighting against harmful mushrooms
- 专利标题（中）： 5-烷基-7-氨基三唑并嘧啶，其生产所需的方法和中间产物，含有所述化合物的试剂及其用于防治有害蘑菇的用途
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申请号： US10531981申请日： 2003-11-04
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公开(公告)号： US20050272749A1公开(公告)日： 2005-12-08
- 发明人: Jordi Tormo Blasco , Carsten Bletner , Bernd Muller , Markus Gewehr , Wassilios Grammenos , Thomas Grote , Andreas Gypser , Joachim Rheinheimer , Peter Schafer , Frank Schieweck , Anja Schwogler , Eberhard Ammermann , Siegfried Strathmann , Ulrich Schofl , Reinhard Stierl
- 申请人： Jordi Tormo Blasco , Carsten Bletner , Bernd Muller , Markus Gewehr , Wassilios Grammenos , Thomas Grote , Andreas Gypser , Joachim Rheinheimer , Peter Schafer , Frank Schieweck , Anja Schwogler , Eberhard Ammermann , Siegfried Strathmann , Ulrich Schofl , Reinhard Stierl
- 申请人地址： DE 67056 Ludwigshafen
- 专利权人： BASF Aktiengesellschaft
- 当前专利权人： BASF Aktiengesellschaft
- 当前专利权人地址： DE 67056 Ludwigshafen
- 优先权： DE10252261.8 20021107
- 国际申请： PCT/EP03/12277 WO 20031104
- 主分类号： C07D487/04
- IPC分类号： C07D487/04 ; A61K31/519
摘要：
5-Alkyl-7-aminotriazolopyrimidines of the formula I, where: R1, R2 are hydrogen, alkyl, alkenyl, alkynyl, haloalkyl, cycloalkyl, phenyl, naphthyl; 5- or 6-membered saturated, unsaturated or aromatic heterocyclyl which contains one to four nitrogen atoms or one to three nitrogen atoms and one sulfur or oxygen atom; or R1 and R2 together with the bridging nitrogen atom can form a 5- or 6-membered ring which contains one to four nitrogen atoms or one to three nitrogen atoms and one sulfur or oxygen atom; R3 is cycloalkyl or bicycloalkyl; where R1, R2 and R3 may be substituted as outlined in the description; X is alkyl or haloalkyl; and their salts; processes and intermediates for their preparation, compositions comprising them and their use for controlling phytopathogenic harmful fungi are described.