发明申请
US20060004002A1 Small molecule thienopyrimidine-based protein tyrosine kinase inhibitors
审中-公开
小分子噻吩并嘧啶类蛋白酪氨酸激酶抑制剂
- 专利标题: Small molecule thienopyrimidine-based protein tyrosine kinase inhibitors
- 专利标题(中): 小分子噻吩并嘧啶类蛋白酪氨酸激酶抑制剂
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申请号: US10884224申请日: 2004-07-02
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公开(公告)号: US20060004002A1公开(公告)日: 2006-01-05
- 发明人: Thomas Thrash , Larry Cabell , Daniel Lohse , Raymond Budde
- 申请人: Thomas Thrash , Larry Cabell , Daniel Lohse , Raymond Budde
- 主分类号: A61K31/5377
- IPC分类号: A61K31/5377 ; A61K31/519 ; C07D515/04
摘要:
Various thienopyrimidine-based analog compounds are able to selectively inhibit the Src family of tyrosine kinases. These compounds are useful in the treatment of various diseases including hyperproliferative diseases, hematologic diseases, osteoporosis, neurological diseases, autoimmune diseases, allergic/immunological diseases, or viral infections.