发明申请
- 专利标题: THERAPEUTIC USES OF DERIVATIVES OF PIPERIDINYL- AND PIPERAZINYL-ALKYL CARBAMATES
- 专利标题(中): 哌啶基和哌嗪酸亚胺衍生物的治疗用途
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申请号: US11670690申请日: 2007-02-02
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公开(公告)号: US20070142350A1公开(公告)日: 2007-06-21
- 发明人: Ahmed ABOUABDELLAH , Philippe BURNIER , Christian HOORNAERT , Jean JEUNESSE , Frederic PUECH
- 申请人: Ahmed ABOUABDELLAH , Philippe BURNIER , Christian HOORNAERT , Jean JEUNESSE , Frederic PUECH
- 申请人地址: FR Paris
- 专利权人: SANOFI-AVENTIS
- 当前专利权人: SANOFI-AVENTIS
- 当前专利权人地址: FR Paris
- 优先权: FR0305540 20030507
- 主分类号: A61K31/53
- IPC分类号: A61K31/53 ; A61K31/519 ; A61K31/517 ; A61K31/506 ; A61K31/4745 ; A61K31/4743 ; A61K31/4741 ; A61K31/497 ; A61K31/501
摘要:
Therapeutic uses of a compound corresponding to the general formula (I): in which A=N or CR2; R2=H, F, OH, CN, CF3, C1-6-alkyl, C1-6-alkoxy; n=2 or 3 and m=2 when A=N; n=1, 2 or 3 and m=1 or 2 when A=CR2; B=covalent bond or C1-8-alkylene; R1=optionally substituted heteroaryl; R3=CHR4CONHR5; R4=H or C1-6-alkyl; R5=H, C1-6-alkyl, C3-7-cycloalkyl, C3-7-cycloalkyl-C1-C6-alkylene; in the form of a base, an acid-addition salt, a hydrate or a solvate.