发明申请
- 专利标题： Processes For The Preparation Of Optically Active Intermediates
- 专利标题（中）： 光学活性中间体的制备方法
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申请号： US11833266申请日： 2007-08-03
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公开(公告)号： US20080071114A1公开(公告)日： 2008-03-20
- 发明人: Masaru Mitsuda , Tadashi Moroshima , Kentaro Tsukuya , Kazuhiko Watabe , Masahiko Yamada
- 申请人： Masaru Mitsuda , Tadashi Moroshima , Kentaro Tsukuya , Kazuhiko Watabe , Masahiko Yamada
- 申请人地址： SE Sodertalje
- 专利权人： ASTRAZENECA AB
- 当前专利权人： ASTRAZENECA AB
- 当前专利权人地址： SE Sodertalje
- 优先权： GB0615620.2 20060805
- 主分类号： C07C209/00
- IPC分类号： C07C209/00
摘要：
This invention relates to processes for the production of optically active 2-(disubstituted aryl)cyclopropylamine compounds and optically active 2-(disubstituted aryl)cyclopropane carboxamide compounds which are useful intermediates for the preparation of pharmaceutical agents, and in particular the compound [1S-(1α,2α,3β(1S*,2R*),5β)]-3-[7-[2-(3,4-difluorophenyl)-cyclopropyl]amino]-5-(propylthio)-3H-1,2,3-triazolo[4,5-d]pyrimidin-3-yl)-5-(2-hydroxyethoxy)-cyclopentane-1,2-diol.
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