发明申请
US20090137573A1 1,3-Disubstituted 4-methyl-1H-pyrrole-2-carboxamides and their Use in Medicaments
有权
1,3-二取代的4-甲基-1H-吡咯-2-甲酰胺及其在药物中的用途
- 专利标题： 1,3-Disubstituted 4-methyl-1H-pyrrole-2-carboxamides and their Use in Medicaments
- 专利标题（中）： 1,3-二取代的4-甲基-1H-吡咯-2-甲酰胺及其在药物中的用途
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申请号： US12331011申请日： 2008-12-09
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公开(公告)号： US20090137573A1公开(公告)日： 2009-05-28
- 发明人: Stefan Oberboersch , Bernd Sundermann , Corinna Sundermann , Edward Bijsterveld , Hagen-Heinrich Hennies
- 申请人： Stefan Oberboersch , Bernd Sundermann , Corinna Sundermann , Edward Bijsterveld , Hagen-Heinrich Hennies
- 申请人地址： DE Aachen
- 专利权人： Gruenenthal GmbH
- 当前专利权人： Gruenenthal GmbH
- 当前专利权人地址： DE Aachen
- 优先权： DE102006027229 20060609
- 主分类号： A61K31/541
- IPC分类号： A61K31/541 ; C07D417/02 ; A61K31/433 ; A61K31/5377 ; A61P25/00 ; C07D413/02 ; C07D295/14 ; A61K31/40
摘要：
1,3-disubstituted 4-methyl-1H-pyrrole-2-carboxamides corresponding to formula I methods for their production, pharmaceutical compositions containing them, and the use thereof for noradrenalin receptor regulation, particularly for inhibiting noradrenalin reuptake, and/or for 5-HT receptor regulation, particularly for inhibiting 5-hydroxy tryptophan reuptake, and/or for opioid receptor regulation and/or for batrachotoxin (BTX) receptor regulation and/or for treating or inhibiting pain and other conditions.
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