发明申请
- 专利标题: CLASS OF HISTONE DEACETYLASE INHIBITORS
- 专利标题(中): 类固醇脱乙酰酶抑制剂
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申请号: US12295498申请日: 2007-03-30
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公开(公告)号: US20100113438A1公开(公告)日: 2010-05-06
- 发明人: Antonello Mai , Saverio Minucci , Florian Thaler , Gilles Pain , Andrea Colombo , Stefania Gagliardi
- 申请人: Antonello Mai , Saverio Minucci , Florian Thaler , Gilles Pain , Andrea Colombo , Stefania Gagliardi
- 申请人地址: IT Milano
- 专利权人: DAC S.R.L.
- 当前专利权人: DAC S.R.L.
- 当前专利权人地址: IT Milano
- 优先权: ITMI2006A000621 20060331
- 国际申请: PCT/EP07/53097 WO 20070330
- 主分类号: A61K31/535
- IPC分类号: A61K31/535 ; C07D401/10 ; A61K31/497 ; A61K31/4545 ; C07D265/30
摘要:
New histone deacetylase inhibitors according to the general formula (I) wherein: Q is a bond, CH2, CH—NR3R4, NR5 or oxygen, X is CH or nitrogen, Y is a bond, CH2, oxygen or NR6, Z is CH or nitrogen, R1, R2 are, independently, hydrogen, halogen, C1-C6 alkyl or C1-C6 haloalkyl, R11, R12 are, independently, hydrogen or C1-C6 alkyl, and R3, R4, R5 and R6 are as further defined in the specification.