利索-全球专利检索

  1. 登录
  2. 注册
发明申请
US20100240717A1 NOVEL THIOPHENE DERIVATIVES AS S1P1/EDG1 RECEPTOR AGONISTS 有权
新型的THIOPHENE衍生物作为S1P1 / EDG1受体激动剂

NOVEL THIOPHENE DERIVATIVES AS S1P1/EDG1 RECEPTOR AGONISTS
摘要：
The invention relates to thiophene derivatives of formula (I)/their preparation and their use as pharmaceutically active compounds. Said compounds particularly act as immunosuppressive agents wherein: A represents *—CO—CH═CH—, *—CO—CH2CH2—, *—CO—CH2—NH—, wherein the sterisks indicate the bond that is linked to the thiophene group of Formula (I), and R1-R3 are as defined in the claims.
摘要（中）：

本发明涉及式（I）的噻吩衍生物/其制备及其作为药物活性化合物的用途。 所述化合物特别充当免疫抑制剂，其中：A表示* -CO-CH = CH-，* -CO-CH 2 CH 2 - ，* -CO-CH 2 -NH-，其中所述甾体表示与噻吩基团连接的键 式（I）和R 1 -R 3如权利要求中所定义。

公开/授权文献
信息查询
Global Dossier Espacenet
0/0