发明申请
US20110060145A1 PROCESS FOR PRODUCTION OF COMPOUND HAVING ANTAGONISTIC ACTIVITY ON NPYY5 RECEPTOR, AND USEFUL CRYSTAL
审中-公开
生产具有NPYY5受体拮抗活性的化合物的方法和有用的晶体
- 专利标题： PROCESS FOR PRODUCTION OF COMPOUND HAVING ANTAGONISTIC ACTIVITY ON NPYY5 RECEPTOR, AND USEFUL CRYSTAL
- 专利标题（中）： 生产具有NPYY5受体拮抗活性的化合物的方法和有用的晶体
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申请号： US12990782申请日： 2009-05-07
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公开(公告)号： US20110060145A1公开(公告)日： 2011-03-10
- 发明人: Yoshihide Sugata , Yutaka Ide , Teruo Sakata , Sohei Omura
- 申请人： Yoshihide Sugata , Yutaka Ide , Teruo Sakata , Sohei Omura
- 申请人地址： JP Osaka-Shi, Osaka
- 专利权人： Shionogi & Co., Ltd.
- 当前专利权人： Shionogi & Co., Ltd.
- 当前专利权人地址： JP Osaka-Shi, Osaka
- 优先权： JP2008-122154 20080508
- 国际申请： PCT/JP2009/058608 WO 20090507
- 主分类号： C07D211/72
- IPC分类号： C07D211/72
摘要：
Disclosed are process for producing a compound having NPYY5 receptor antagonism and useful crystals.A process for producing a compound represented by the formula (IV): wherein R1 is substituted or unsubstituted alkyl, R2 is substituted or unsubstituted alkyl, and n is 1 or 2, or the like, which comprises reacting a compound represented by the formula (II): wherein R1 and n are as defined above, and X is a leaving group, or the like and a compound represented by formula (III): wherein R2 is as defined above, or the like.
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