发明申请
US20110152464A1 PIPECOLIC LINKER AND ITS USE FOR CHEMISTRY ON SOLID SUPPORT
有权
PIPECOLIC连接器及其在固体支持下的化学物质使用
- 专利标题: PIPECOLIC LINKER AND ITS USE FOR CHEMISTRY ON SOLID SUPPORT
- 专利标题(中): PIPECOLIC连接器及其在固体支持下的化学物质使用
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申请号: US13061080申请日: 2009-08-28
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公开(公告)号: US20110152464A1公开(公告)日: 2011-06-23
- 发明人: Jean Martinez , Pawel Zajdel , Maciej Pawlowski , Gilles Subra
- 申请人: Jean Martinez , Pawel Zajdel , Maciej Pawlowski , Gilles Subra
- 申请人地址: FR Montpellier
- 专利权人: UNIVERSITE DE MONTPELLIER I
- 当前专利权人: UNIVERSITE DE MONTPELLIER I
- 当前专利权人地址: FR Montpellier
- 优先权: EP08305512.9 20080829
- 国际申请: PCT/EP2009/061171 WO 20090828
- 主分类号: C08F12/28
- IPC分类号: C08F12/28 ; C07D211/60 ; C07K1/10
摘要:
The present invention relates to a pipecolic linker and its use as a solid-phase linker in organic synthesis. Said pipecolic solid-phase linker may be used for coupling functional groups chosen between primary amines, secondary amines, aromatic amines, alcohols, phenols and thiols. In particular, said pipecolic solid-phase linker may be used for peptide or pseudopeptide synthesis, such as the reverse N to C peptide synthesis or the retro-inverso peptide synthesis, or for the synthesis of small organic molecules.
公开/授权文献
- US08546533B2 Pipecolic linker and its use for chemistry on solid support 公开/授权日:2013-10-01
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