发明申请
US20110178140A1 SULFUR CONTAINING PYRAZOLE-HETEROCYCLE DERIVATIVES AS CANNABINOID CB1 RECEPTOR ANTAGONISTS
失效
作为CANNABINOID CB1受体拮抗剂的含硫吡唑杂交衍生物
- 专利标题： SULFUR CONTAINING PYRAZOLE-HETEROCYCLE DERIVATIVES AS CANNABINOID CB1 RECEPTOR ANTAGONISTS
- 专利标题（中）： 作为CANNABINOID CB1受体拮抗剂的含硫吡唑杂交衍生物
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申请号： US13120026申请日： 2008-09-25
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公开(公告)号： US20110178140A1公开(公告)日： 2011-07-21
- 发明人: Jinhwa Lee , Hee Jeong Seo , Min-Ah Kim , Jeongmin Kim , Sung-Han Lee , Myung Eun Jung , Mi-Soon Kim
- 申请人： Jinhwa Lee , Hee Jeong Seo , Min-Ah Kim , Jeongmin Kim , Sung-Han Lee , Myung Eun Jung , Mi-Soon Kim
- 申请人地址： KR Yongin-si, Gyeonggi-do
- 专利权人： GREEN CROSS CORPORATION
- 当前专利权人： GREEN CROSS CORPORATION
- 当前专利权人地址： KR Yongin-si, Gyeonggi-do
- 国际申请： PCT/KR2008/005689 WO 20080925
- 主分类号： A61K31/433
- IPC分类号： A61K31/433 ; C07D417/04 ; C07D413/04 ; A61K31/4245 ; A61P3/04
摘要：
A novel sulfur containing heteroaryl-pyrazole compound of formula (I) or a pharmaceutically acceptable salt thereof is effective as a cannabinoid CB1 receptor inverse agonist or antagonist, which is useful for preventing or treating obesity and obesity-related metabolic disorders. The prevention also provide a method for preparing same, a pharmaceutical composition containing same, and a method for preventing or treating obesity and obesity-related metabolic disorders.
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