发明申请
- 专利标题： DIPEPTOID PRODRUGS AND THE USE THEREOF
- 专利标题（中）： DIPEPTOID PRODRUGS及其使用
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申请号： US13132991申请日： 2009-12-03
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公开(公告)号： US20110294719A1公开(公告)日： 2011-12-01
- 发明人: Hans-Georg Lerchen , Daniel Meibom , Alexandros Vakalopoulos , Barbara Albrecht-Küpper , Joerg Keldenich , Katja Zimmermann , Peter Nell , Ursula Krenz
- 申请人： Hans-Georg Lerchen , Daniel Meibom , Alexandros Vakalopoulos , Barbara Albrecht-Küpper , Joerg Keldenich , Katja Zimmermann , Peter Nell , Ursula Krenz
- 专利权人： BAYER SCHERING PHARMA
- 当前专利权人： BAYER SCHERING PHARMA
- 优先权： DE102008062567.1 20081216
- 国际申请： PCT/EP09/08617 WO 20091203
- 主分类号： A61K38/05
- IPC分类号： A61K38/05 ; A61P9/10 ; A61P9/00 ; C07K17/02 ; C07K1/04
摘要：
The present application relates to dipeptide-like prodrug derivatives of 2-amino-6-({[2-(4-chlorophenyl)-1,3-oxazol-4-yl]methyl}sulfanyl)-4-(4-{[2,3-dihydroxypropyl]oxy}phenyl)pyridine-3,5-dicarbonitrile, processes for their preparation, their use for the treatment and/or prophylaxis of diseases, and their use for the manufacture of medicaments for the treatment and/or prophylaxis of diseases, especially of cardiovascular disorders.
公开/授权文献
- US08741834B2 Dipeptoid prodrugs and the use thereof 公开/授权日：2014-06-03