发明申请
- 专利标题： TRI-CYCLIC PYRAZOLOPYRIDINE KINASE INHIBITORS
- 专利标题（中）： 三环吡嗪类激酶抑制剂
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申请号： US13216606申请日： 2011-08-24
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公开(公告)号： US20120053187A1公开(公告)日： 2012-03-01
- 发明人: Alex Aronov , Jon H. Come , Kevin Michael Cottrell , Arnaud Le Tiran , Valerie Marone , Gabriel Martinez Botella , David Messersmith , Emilie Porter Huck , Ronald Lee Grey, JR.
- 申请人： Alex Aronov , Jon H. Come , Kevin Michael Cottrell , Arnaud Le Tiran , Valerie Marone , Gabriel Martinez Botella , David Messersmith , Emilie Porter Huck , Ronald Lee Grey, JR.
- 申请人地址： US MA Cambridge
- 专利权人： VERTEX PHARMACEUTICALS INCORPORATED
- 当前专利权人： VERTEX PHARMACEUTICALS INCORPORATED
- 当前专利权人地址： US MA Cambridge
- 主分类号： A61K31/444
- IPC分类号： A61K31/444 ; A61K31/497 ; C07D417/14 ; C12N9/99 ; A61P25/00 ; A61P29/00 ; A61P37/02 ; A61P37/06 ; C07D401/14 ; A61K31/4439
摘要：
The present invention relates to compounds useful as inhibitors of PI3K, particularly of PI3Kγ. The invention also provides pharmaceutically acceptable compositions comprising said compounds and methods of using the compositions in the treatment of various disease, conditions, or disorders.
公开/授权文献
- US08268999B2 Tri-cyclic pyrazolopyridine kinase inhibitors 公开/授权日：2012-09-18