发明申请
- 专利标题： PICOLINAMIDE DERIVATIVES AS TTX-S BLOCKERS
- 专利标题（中）： PICOLINAMIDE衍生物作为TTX-S阻断剂
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申请号： US13388740申请日： 2010-08-04
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公开(公告)号： US20120142691A1公开(公告)日： 2012-06-07
- 发明人: Hirohide Noguchi , Tadashi Inoue , Mikio Morita , Yoshimasa Arano
- 申请人： Hirohide Noguchi , Tadashi Inoue , Mikio Morita , Yoshimasa Arano
- 专利权人： RAQUALIA PHARMA INC.
- 当前专利权人： RAQUALIA PHARMA INC.
- 国际申请： PCT/JP2010/004917 WO 20100804
- 主分类号： A61K31/5377
- IPC分类号： A61K31/5377 ; C07D401/14 ; C07D413/14 ; A61K31/4439 ; A61K31/444 ; A61K31/4545 ; A61P1/00 ; A61P25/00 ; A61P19/08 ; A61P19/02 ; A61P1/18 ; A61P25/08 ; A61P9/06 ; A61P25/22 ; A61P25/24 ; A61P5/00 ; A61P29/00 ; C07D401/12
摘要：
The present invention relates to picolinamide derivatives which have blocking activities of voltage gated sodium channels as the TTX-S channels, and which are useful in the treatment or prevention of disorders and diseases in which voltage gated sodium channels are involved. The invention also relates to pharmaceutical compositions comprising these compounds and the use of these compounds and compositions in the prevention or treatment of such diseases in which voltage gated sodium channels are involved.
公开/授权文献
- US08809380B2 Picolinamide derivatives as TTX-S blockers 公开/授权日：2014-08-19
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