发明申请
US20120178904A1 PEPTIDE ANALOGS THAT ARE POTENT AND SELECTIVE FOR HUMAN NEUROTENSIN RECEPTOR SUBTYPE 2
审中-公开
对于人神经递质受体亚型2的肽类型和选择性
- 专利标题： PEPTIDE ANALOGS THAT ARE POTENT AND SELECTIVE FOR HUMAN NEUROTENSIN RECEPTOR SUBTYPE 2
- 专利标题（中）： 对于人神经递质受体亚型2的肽类型和选择性
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申请号： US13177909申请日： 2011-07-07
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公开(公告)号： US20120178904A1公开(公告)日： 2012-07-12
- 发明人: Elliot RICHELSON , Daniel J. McCORMICK , Yuan-Ping PANG , Kenneth S. PHILLIPS
- 申请人： Elliot RICHELSON , Daniel J. McCORMICK , Yuan-Ping PANG , Kenneth S. PHILLIPS
- 主分类号： C07K7/06
- IPC分类号： C07K7/06
摘要：
Neurotensin analogs selective for neurotensin receptor subtype 2 are described. These include hexapeptides (NT(8-13)) and pentapeptides (NT(9-13)) having a D-3,1-naphthyl-alanine, D-3,2-naphthyl-alanine, an alanine derivative such as cyclohexylalanine, or 1,2,3,4-tetrahydroisoquinoline at position 11. Methods of treating pain by administering these neurotensin analogs are also described.
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