发明申请
US20130096094A1 Derivatives of 3-O-(3',3'-dimethylsuccinyl)-betulinic acid
有权
3-O-（3'，3'-二甲基琥珀酰基） - 丁酰酸的衍生物
- 专利标题： Derivatives of 3-O-(3',3'-dimethylsuccinyl)-betulinic acid
- 专利标题（中）： 3-O-（3'，3'-二甲基琥珀酰基） - 丁酰酸的衍生物
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申请号： US13608486申请日： 2012-09-10
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公开(公告)号： US20130096094A1公开(公告)日： 2013-04-18
- 发明人: Serge Bouaziz , Pascale Coric , Pierre Boulanger , Saw-See Hong , Serge Turcaud , Florence Souquet , Nathalie Chazal , Laurence Briant
- 申请人： Serge Bouaziz , Pascale Coric , Pierre Boulanger , Saw-See Hong , Serge Turcaud , Florence Souquet , Nathalie Chazal , Laurence Briant
- 申请人地址： FR Paris FR Paris
- 专利权人： Universite Paris Descartes,Centre National de la Recherche Scientifique
- 当前专利权人： Universite Paris Descartes,Centre National de la Recherche Scientifique
- 当前专利权人地址： FR Paris FR Paris
- 优先权： EP11306138.6 20110912
- 主分类号： C07J53/00
- IPC分类号： C07J53/00
摘要：
The present invention relates to compounds of the following formula (I): or a pharmaceutically acceptable salt thereof, a stereoisomer or a mixture of stereoisomers in any proportion, in particular a mixture of enantiomers, and particularly a racemate mixture, in which R represents a (C1-C10)alkyl group substituted with one or more, preferably one or two, groups chosen from COOH and NHR1, with R1 representing a hydrogen atom or a -Alk, —C(O)-Alk or —C(O)O-Alk group, Alk representing a (C1-C6)alkyl group, as well as a method for preparing them, and their use as a medicine, notably for treating an infection with a retrovirus such as HIV.
公开/授权文献
- US09056888B2 Derivatives of 3-O-(3',3'-dimethylsuccinyl)-betulinic acid 公开/授权日：2015-06-16
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