- 专利标题: NOVEL SOLID FORMS OF TACEDINALINE
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申请号: US13620761申请日: 2012-09-15
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公开(公告)号: US20130150450A1公开(公告)日: 2013-06-13
- 发明人: Edward Holson , Florence F. Wagner , G. Patrick Stahly
- 申请人: Edward Holson , Florence F. Wagner , G. Patrick Stahly
- 申请人地址: US MA Cambridge
- 专利权人: THE BROAD INSTITUTE, INC.
- 当前专利权人: THE BROAD INSTITUTE, INC.
- 当前专利权人地址: US MA Cambridge
- 主分类号: C07C233/80
- IPC分类号: C07C233/80
摘要:
Novel solid forms of tacedinaline (4-(acetylamino)-N-(2-aminophenyl)benzamide), including crystalline tacedinaline Forms A, B, and D, a novel crystalline tacedinaline TFA salt, and amorphous tacedinaline, are disclosed. Pharmaceutical compositions comprising crystalline tacedinaline Forms A, B, and D, the novel crystalline tacedinaline TFA salt, and/or amorphous tacedinaline, and methods of treating various conditions by administering those novel solid forms, are also disclosed.
公开/授权文献
- US08729130B2 Methods of using novel solid forms of tacedinaline 公开/授权日:2014-05-20