发明申请
- 专利标题: New Process for the Preparation of Aryl Substituted Olefinic Amines
- 专利标题(中): 制备芳基取代的烯属胺的新方法
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申请号: US13697807申请日: 2011-05-19
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公开(公告)号: US20130225827A1公开(公告)日: 2013-08-29
- 发明人: Gary Maurice Dull , John Genus , Tommi Ratilainen , Per Olof Ryberg , Janna Hellstrom , Niklas Wahlstrom , Thomas Wannman
- 申请人: Gary Maurice Dull , John Genus , Tommi Ratilainen , Per Olof Ryberg , Janna Hellstrom , Niklas Wahlstrom , Thomas Wannman
- 申请人地址: US NC Winston-Salem SE Sodertalje
- 专利权人: TARGACEPT, INC.,ASTRAZENECA AB
- 当前专利权人: TARGACEPT, INC.,ASTRAZENECA AB
- 当前专利权人地址: US NC Winston-Salem SE Sodertalje
- 国际申请: PCT/SE2011/050630 WO 20110519
- 主分类号: C07D213/65
- IPC分类号: C07D213/65 ; C07C211/21
摘要:
An improved process for the preparation of aryl substituted olefinic amines such as (2S)-(4E)-N-methyl-5-[3-(5-isopropoxypyridin)yl]-4-penten-2-amine and (2S)-(4E)-N-methyl-5-[3-(5-methoxypyridin)yl]-4-penten-2-amine and new intermediates used in said process.