Invention Application
US20160002165A1 SALT OF PYRROLIDIN-3-YL ACETIC ACID DERIVATIVE AND CRYSTALS THEREOF 有权
吡咯烷-3-基乙酸衍生物及其结晶盐

  • Patent Title: SALT OF PYRROLIDIN-3-YL ACETIC ACID DERIVATIVE AND CRYSTALS THEREOF
  • Patent Title (中): 吡咯烷-3-基乙酸衍生物及其结晶盐
  • Application No.: US14768520
    Application Date: 2014-03-10
  • Publication No.: US20160002165A1
    Publication Date: 2016-01-07
  • Inventor: Kenshi YoshidaIkuo Kushida
  • Applicant: EISAI R&D MANAGEMENT CO., LTD.
  • Priority: JP2013-049619 20130312
  • International Application: PCT/JP2014/056123 WO 20140310
  • Main IPC: C07D211/58
  • IPC: C07D211/58 C07C59/50
SALT OF PYRROLIDIN-3-YL ACETIC ACID DERIVATIVE AND CRYSTALS THEREOF
Abstract:
An organic carboxylic acid salt of 2-[(3S,4R)-1-{[2-chloro-6-(trifluoromethyl)phenyl]methyl}-3-{[1-(cyclohex-1-en-1-ylmethyl) piperidin-4-yl]carbamoyl}-4-methylpyrrolidin-3-yl]acetic acid and a crystal thereof.
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