发明申请
US20160207918A1 SUBSTITUTED AZAINDOLEOXOACETIC PIPERAZINE DERIVATIVES WITH PROTEASE
INHIBITORS
审中-公开
带有蛋白酶抑制剂的取代的氮杂双环戊哌嗪衍生物
- 专利标题： SUBSTITUTED AZAINDOLEOXOACETIC PIPERAZINE DERIVATIVES WITH PROTEASE INHIBITORS
- 专利标题（中）： 带有蛋白酶抑制剂的取代的氮杂双环戊哌嗪衍生物
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申请号： US15071329申请日： 2016-03-16
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公开(公告)号： US20160207918A1公开(公告)日： 2016-07-21
- 发明人: Tao Wang , Zhongxing Zhang , Nicholas A. Meanwell , John F. Kadow , Zhiwei Yin , Qiufen May Xue , Alicia Regueiro-Ren , John D. Matiskella , Yasutsugu Ueda
- 申请人： BRISTOL-MYERS SQUIBB COMPANY
- 主分类号： C07D471/04
- IPC分类号： C07D471/04 ; C07D491/048
摘要：
This invention provides compounds having drug and bio-affecting properties, their pharmaceutical compositions and method of use. In particular, the invention is concerned with azaindoleoxoacetyl piperazine derivatives having the Formula I: wherein Q is These compounds possess unique antiviral activity, whether used alone or in combination with other antivirals, antiinfectives, immunomodulators or HIV entry inhibitors. More particularly, the present invention relates to the treatment of HIV and AIDS.
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