Invention Application
- Patent Title: CRYSTALLINE FORMS OF PARP INHIBITORS
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Application No.: US15529883Application Date: 2015-11-25
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Publication No.: US20170267683A1Publication Date: 2017-09-21
- Inventor: Stephen J. BIERLMAIER , Ralph C. HALTIWANGER , Martin J. JACOBS
- Applicant: CEPHALON, INC.
- Applicant Address: US PA Frazer
- Assignee: CEPHALON, INC.
- Current Assignee: CEPHALON, INC.
- Current Assignee Address: US PA Frazer
- International Application: PCT/US2015/062572 WO 20151125
- Main IPC: C07D487/04
- IPC: C07D487/04 ; C07C57/15 ; C07C59/245 ; C07D207/28 ; C07C59/06 ; C07C53/10

Abstract:
The present disclosure relates to crystalline forms of 4,5,6,7-tetrahydro-11-methoxy-2-[(4-methyl-1-piperazinyl)methyl]-1H-cyclopenta[a]pyrrolo[3,4-c]carbazole-1,3(2H)-dione, including salts forms and free base forms.
Public/Granted literature
- US10150772B2 Crystalline forms of PARP inhibitors Public/Granted day:2018-12-11
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