NOVEL INTERMEDIATES USEFUL FOR THE SYNTHESIS OF AMINOPYRIMIDINE DERIVATIVES, PROCESS FOR PREPARING THE SAME, AND PROCESS FOR PREPARING AMINOPYRIMIDINE DERIVATIVES USING THE SAME

发明申请

US20200207750A1 NOVEL INTERMEDIATES USEFUL FOR THE SYNTHESIS OF AMINOPYRIMIDINE DERIVATIVES, PROCESS FOR PREPARING THE SAME, AND PROCESS FOR PREPARING AMINOPYRIMIDINE DERIVATIVES USING THE SAME 审中-公开

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专利标题： NOVEL INTERMEDIATES USEFUL FOR THE SYNTHESIS OF AMINOPYRIMIDINE DERIVATIVES, PROCESS FOR PREPARING THE SAME, AND PROCESS FOR PREPARING AMINOPYRIMIDINE DERIVATIVES USING THE SAME
申请号： US16633695

申请日： 2018-07-25
公开(公告)号： US20200207750A1

公开(公告)日： 2020-07-02
发明人: Sang-Ho OH , Ja-Heouk KHOO , Jong-Chul LIM , Doo-Byung LEE , Jung-Ae LEE , Jun-Sup LEE , Hyun JU , Woo-Seob SHIN , Sang-Seol JEON
申请人： Yuhan Corporation
优先权： com.zzzhc.datahub.patent.etl.us.BibliographicData$PriorityClaim@a0ccf86
国际申请： PCT/KR2018/008381 WO 20180725
主分类号： C07D413/14
IPC分类号： C07D413/14 ; C07D265/32 ; C07D403/10

NOVEL INTERMEDIATES USEFUL FOR THE SYNTHESIS OF AMINOPYRIMIDINE DERIVATIVES, PROCESS FOR PREPARING THE SAME, AND PROCESS FOR PREPARING AMINOPYRIMIDINE DERIVATIVES USING THE SAME

摘要：

The present invention provides a novel process for preparing an aminopyrimidine derivative or pharmaceutically acceptable salt thereof having a selective inhibitory activity against protein kinases, especially against the protein kinases for mutant epidermal growth factor receptors. And also, the present invention provides novel intermediates useful for said process and processes for preparing the same.

公开/授权文献

US10858353B2 Intermediates useful for the synthesis of aminopyrimidine derivatives, process for preparing the same, and process for preparing aminopyrimidine derivatives using the same 公开/授权日：2020-12-08

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IPC分类:

C	化学；冶金
C07	有机化学
C07D	杂环化合物（高分子化合物入C08）
C07D413/00	杂环化合物，含两个或更多个杂环，至少有1个环有氮原子和氧原子作为仅有的杂环原子
C07D413/14	.含有3个或更多个杂环