发明授权
US4503075A Derivatives of
1-alkylamine-3[4(p-alkyloxy-benzamide)phenoxy]-2-propanol, having
beta-sympatholytic activity, their salts, and production processes
thereof
失效
具有β-交替溶解活性的1-烷基胺-3 [4（对 - 烷氧基 - 苯甲酰胺）苯氧基] -2-丙醇的衍生物及其盐及其制备方法
- 专利标题： Derivatives of 1-alkylamine-3[4(p-alkyloxy-benzamide)phenoxy]-2-propanol, having beta-sympatholytic activity, their salts, and production processes thereof
- 专利标题（中）： 具有β-交替溶解活性的1-烷基胺-3 [4（对 - 烷氧基 - 苯甲酰胺）苯氧基] -2-丙醇的衍生物及其盐及其制备方法
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申请号： US441101申请日： 1982-11-12
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公开(公告)号： US4503075A公开(公告)日： 1985-03-05
- 发明人: Vittorio Pestellini , Mario Ghelardoni , Danilo Giannotti , Alessandro Giolitti , Carlo A. Maggi , Stefano Manzini , Guglielmo Grimaldi , Alberto Meli
- 申请人： Vittorio Pestellini , Mario Ghelardoni , Danilo Giannotti , Alessandro Giolitti , Carlo A. Maggi , Stefano Manzini , Guglielmo Grimaldi , Alberto Meli
- 申请人地址： ITX
- 专利权人： A. Menarini S.A.S.
- 当前专利权人： A. Menarini S.A.S.
- 当前专利权人地址： ITX
- 主分类号： A61K31/165
- IPC分类号： A61K31/165 ; C07C233/12 ; C07C103/82
摘要：
The invention comprises: a derivative of 1-alkylamine-3-[4(p-alkyloxy-benzamide)phenoxy]-2-propanol of general formula I: ##STR1## where R.sub.1 is a linear or branched alkyl chain with 1 to 8 carbon atoms included, an alkenyl chain with 2 to 8 carbon atoms included, or an arylalkyl chain with 7 to 10 carbon atoms included, and R is a linear or branched alkyl group with 1 to 8 carbon atoms included;a compound as above, in an optically active form;pharmaceutically acceptable, non toxic salts of the above compounds;synthesis processes for obtaining the above compounds; anda pharmaceutical composition based on a compound as defined above.
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