发明授权
- 专利标题: Anthelmintics
- 专利标题(中): ANTHELMINTICS
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申请号: US586176申请日: 1990-09-19
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公开(公告)号: US5081125A公开(公告)日: 1992-01-14
- 发明人: Peter Maienfisch , Christor Hildenbrand , Jean-Claude Gehret
- 申请人: Peter Maienfisch , Christor Hildenbrand , Jean-Claude Gehret
- 申请人地址: NY Ardsley
- 专利权人: Ciba-Geigy Corporation
- 当前专利权人: Ciba-Geigy Corporation
- 当前专利权人地址: NY Ardsley
- 优先权: CHX3481/89 19890926
- 主分类号: A23K1/16
- IPC分类号: A23K1/16 ; A61K31/44 ; A61K31/4402 ; A61K31/4418 ; A61K31/505 ; A61P33/00 ; C07D213/64 ; C07D213/643 ; C07D213/70 ; C07D213/84 ; C07D213/85 ; C07D239/34 ; C07D239/38 ; C07D239/56
摘要:
Anthelmintically active compounds of formula I are described ##STR1## in which R.sub.1 is hydrogen, halogen, C.sub.1 -C.sub.2 alkyl, C.sub.1 -C.sub.2 thioalkyl, C.sub.1 -C.sub.2 haloalkyl, nitro, C.sub.1 -C.sub.2 alkoxy, or the group SO.sub.n R in which R is C.sub.1 -C.sub.2 alkyl or phenyl and n is 0, 1 or 2;R.sub.2 is hydrogen, halogen, C.sub.1 -C.sub.2 alkyl, C.sub.1 -C.sub.2 haloalkyl, C.sub.1 -C.sub.2 haloalkoxy or C.sub.1 -C.sub.2 alkoxy;R.sub.3 is hydrogen or C.sub.1 -C.sub.2 alkyl;R.sub.4 is hydrogen or C.sub.1 -C.sub.2 alkyl;R.sub.5 is hydrogen, halogen or C.sub.1 -C.sub.5 alkyl;R.sub.6 is hydrogen, halogen or C.sub.1 -C.sub.5 alkyl;R.sub.7 is hydrogen, halogen, C.sub.1 -C.sub.2 alkyl, nitro, C.sub.1 -C.sub.2 haloalkyl, C.sub.1 -C.sub.2 haloalkoxy or C.sub.1 -C.sub.2 alkoxy;R.sub.8 is hydrogen, halogen, C.sub.1 -C.sub.2 alkyl, C.sub.1 -C.sub.2 haloalkyl, C.sub.1 -C.sub.2 haloalkoxy or C.sub.1 -C.sub.2 alkoxy;R.sub.9 is hydrogen, halogen, C.sub.1 -C.sub.2 alkyl, C.sub.1 -C.sub.2 haloalkyl, C.sub.1 -C.sub.2 haloalkoxy or C.sub.1 -C.sub.2 alkoxy;R.sub.10 is hydrogen, halogen, C.sub.1 -C.sub.6 alkyl, C.sub.1 -C.sub.2 haloalkyl, C.sub.1 -C.sub.2 alkylthio, C.sub.3 -C.sub.6 cycloalkyl or cyano;R.sub.11 is hydrogen, halogen, C.sub.1 -C.sub.6 alkyl, C.sub.1 -C.sub.2 haloalkyl, C.sub.1 -C.sub.2 alkylthio or C.sub.3 -C.sub.6 cycloalkyl;R.sub.12 is hydrogen or halogen; and Y is .dbd.CH-- or .dbd.N-; including the physiologically tolerable acid additon salts thereof, and also the preparatin and use thereof and novel intermediates.
公开/授权文献
- USD282456S Tire 公开/授权日:1986-02-04
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