发明授权
US06187812B1 Phenylacetic acid derivatives, preparation thereof and intermediates therefor, and compositions containing them
失效
苯乙酸衍生物,其制备方法及其中间体,以及含有它们的组合物
- 专利标题: Phenylacetic acid derivatives, preparation thereof and intermediates therefor, and compositions containing them
- 专利标题(中): 苯乙酸衍生物,其制备方法及其中间体,以及含有它们的组合物
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申请号: US09497152申请日: 2000-02-03
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公开(公告)号: US06187812B1公开(公告)日: 2001-02-13
- 发明人: Herbert Bayer , Hubert Sauter , Ruth Müller , Wassilios Grammenos , Albrecht Harreus , Reinhard Kirstgen , Franz Röhl , Eberhard Ammermann , Gisela Lorenz
- 申请人: Herbert Bayer , Hubert Sauter , Ruth Müller , Wassilios Grammenos , Albrecht Harreus , Reinhard Kirstgen , Franz Röhl , Eberhard Ammermann , Gisela Lorenz
- 优先权: DE4403448 19940204; DE4421182 19940617
- 主分类号: A01N3718
- IPC分类号: A01N3718
摘要:
Phenylacetic acid derivatives of the formula I where the substituents and the index have the following meanings: X is oxygen or sulfur; R is hydrogen or alkyl; R1 is hydrogen or alkyl; R2 is cyano, nitro, trifluoromethyl, halogen, alkyl or alkoxy; m is 0, 1 or 2, it being possible for the R2 radicals to be different if m is 2; R3 is hydrogen, cyano, nitro, hydroxyl, amino, halogen, alkyl, haloalkyl, alkoxy, haloalkoxy, alkylthio, alkylamino or dialkylamino; R4 is hydrogen, cyano, nitro, hydroxyl, amino, halogen, unsubstituted or substituted alkyl, alkoxy, alkylthio, alkylamino, dialkylamino, alkenyl, alkenyloxy, alkenylthio, alkenylamino, N-alkenyl-N-alkylamino, alkynyl, alkynyloxy, alkynylthio, alkynylamino, N-alkynyl-N-alkylamino; unsubstituted or substituted cycloalkyl, cycloalkoxy, cycloalkylthio, cycloalkylamino, N-cycloalkyl-N-alkylamino, cycloalkenyl, cycloalkenyloxy, cycloalkenylthio, cycloalkenylamino, N-cycloalkenyl-N-alkylamino, heterocyclyl, heterocyclyloxy, heterocyclylthio, heterocyclylamino, N-heterocyclyl-N-alkylamino, aryl, aryloxy, arylthio, arylamino, N-aryl-N-alkylamino, hetaryl, hetaryloxy, hetarylthio, hetaryl amino, N-hetaryl-N-alkylamino; R5 is hydrogen, unsubstituted or substituted alkyl, cycloalkyl, alkenyl, alkynyl, alkylcarbonyl, alkenylcarbonyl, alkynylcarbonyl or alkylsulfonyl; unsubstituted or substituted aryl, arylcarbonyl, arylsulfonyl; hetaryl, hetarylcarbonyl or hetarylsulfonyl, and their salts, processes and intermediates for their preparation, and their use are described.
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