发明授权
US06316474B1 2-benzyl and 2-heteroaryl benzimidazole NMDA/NR2B antagonists
失效
2-苄基和2-杂芳基苯并咪唑NMDA / NR2B拮抗剂
- 专利标题: 2-benzyl and 2-heteroaryl benzimidazole NMDA/NR2B antagonists
- 专利标题(中): 2-苄基和2-杂芳基苯并咪唑NMDA / NR2B拮抗剂
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申请号: US09696501申请日: 2000-10-25
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公开(公告)号: US06316474B1公开(公告)日: 2001-11-13
- 发明人: John A. McCauley , Cory R. Theberge , Nigel J. Liverton , David A. Claremon , Christopher F. Claiborne
- 申请人: John A. McCauley , Cory R. Theberge , Nigel J. Liverton , David A. Claremon , Christopher F. Claiborne
- 主分类号: A01N4340
- IPC分类号: A01N4340
摘要:
Benzimidazoles, substituted in the 2-position by substituted benzyl groups or heteroaryl groups are effective as NMDA NR2B antagonists and are useful for relieving pain.