发明授权
US06384058B1 2,4,6-trisubstituted pryridines with estrogenic activity and methods for the solid phase synthesis thereof
失效
具有雌激素活性的2,4,6-三取代吡啶并用于其固相合成的方法
- 专利标题： 2,4,6-trisubstituted pryridines with estrogenic activity and methods for the solid phase synthesis thereof
- 专利标题（中）： 具有雌激素活性的2,4,6-三取代吡啶并用于其固相合成的方法
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申请号： US09703519申请日： 2000-11-01
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公开(公告)号： US06384058B1公开(公告)日： 2002-05-07
- 发明人: Chingfan Chiu , Zhilian Tang , John W. Ellingboe
- 申请人： Chingfan Chiu , Zhilian Tang , John W. Ellingboe
- 主分类号： C07D40104
- IPC分类号： C07D40104
摘要：
The present invention relates to novel substituted pyridine compounds of Formula (I) wherein the moiety Z, R1, R2 and R3 are as herein defined, having estrogenic activity, to processes for their preparation, to a combinatorial library and solid phase methods for preparing libraries of the compounds, to utilizing libraries of the compounds for drug discovery, to methods of treatment and to pharmaceutical compositions thereof.