发明授权
- 专利标题: 1,3,4-oxadiazole derivatives and process for producing the same
- 专利标题(中): 1,3,4-恶二唑衍生物及其制备方法
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申请号: US09936331申请日: 2001-12-19
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公开(公告)号: US06534658B1公开(公告)日: 2003-03-18
- 发明人: Tsutomu Kojima , Katsutoshi Hachiya , Kazuyuki Ohmoto
- 申请人: Tsutomu Kojima , Katsutoshi Hachiya , Kazuyuki Ohmoto
- 优先权: JP11-066065 19990312
- 主分类号: C07D27110
- IPC分类号: C07D27110
摘要:
Oxadiazole derivatives represented by formula (I): (wherein R1 represents a hydrogen atom or an amino-protective group; R2, R3, and R4 each independently represents an alkyl group, a cycloalkyl group, a phenyl group which may be substituted, or a 3,4-methylenedioxyphenyl group, or R3 and R4 are taken together to represent a C2-6 alkylene group), a process of producing the same, and a process for producing oxadiazole derivatives represented by formula (II): (wherein all symbols have the same meanings as described above) using the above derivative. According to the invention, the compound represented by formula (II) is produced through fewer steps in a high yield.